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SYM 2081
CAS No. 31137-74-3
SYM 2081( —— )
Catalog No. M33504 CAS No. 31137-74-3
SYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 132 | In Stock |
|
| 5MG | 202 | In Stock |
|
| 10MG | 297 | In Stock |
|
| 25MG | 490 | In Stock |
|
| 50MG | 707 | In Stock |
|
| 100MG | 972 | In Stock |
|
| 500MG | 1944 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSYM 2081
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NoteResearch use only, not for human use.
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Brief DescriptionSYM 2081 is a specific kainate receptor agonist with an IC50 value of 35 nM for [3H]-kainate binding. SYM 2081 depolarizes the muscle and reduces the EPSP amplitude.
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DescriptionSYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetiGluR
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RecptoriGluR
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Research Area——
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Indication——
Chemical Information
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CAS Number31137-74-3
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Formula Weight161.16
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Molecular FormulaC6H11NO4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?H2O : 50 mg/mL (310.25 mM; Ultrasonic)
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SMILES[C@@H](C[C@@H](C(O)=O)N)(C(O)=O)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Lee JY, et al. Furthering pharmacological and physiological assessment of the glutamatergic receptors at the Drosophila neuromuscular junction. Comp Biochem Physiol C Toxicol Pharmacol. 2009 Nov;150(4):546-57.?
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